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Limited evidencePhysical performance

Guanidinoacetic Acid (GAA)

The body's direct precursor to creatine. It does raise tissue creatine, but it also raises homocysteine, and it has never been shown to beat simply taking creatine.

Evidence last reviewed: August 2026

What the science says

  • Raises muscle and brain creatine Limited evidence

    A randomised superiority pilot trial in healthy men found guanidinoacetic acid increased muscle and brain creatine more than creatine monohydrate over several weeks. It was a pilot with very few participants.

  • Raises homocysteine Moderate evidence

    A randomised, double-blind trial comparing guanidinoacetic acid plus creatine with creatine alone found the GAA arm developed higher plasma homocysteine, an unwanted change, without a clear performance advantage.

  • No performance case over creatine Limited evidence

    No trial has shown guanidinoacetic acid outperforms creatine monohydrate for exercise performance, and human data cover only weeks to a few months.

Dosage & safety

Studied doseTrials used 1.2–3 g/day for 4–8 weeks, sometimes with creatine and with B vitamins intended to blunt the homocysteine rise.
SafetyIt raises homocysteine; co-supplementation with folate and B12 is proposed but not proven to solve this. Long-term safety is unknown and it is not an authorised novel food in some jurisdictions. Avoid in pregnancy and in kidney disease.

Scientific references

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